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Access to Galectin3 Inhibitors from Chemoenzymatic Synthons

Christophe Dussouy , Stéphane Téletchéa , Annie Lambert , Cathy Charlier , Iuliana Botez , et al.
Journal of Organic Chemistry, 2020, ⟨10.1021/acs.joc.0c01927⟩
Journal articles hal-03010455v1
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Synergetic anticancer activity of gold porphyrin appended to phenyl tin malonate organometallic complexes

Christophe Nguyen , Isabelle Toubia , Stéphane Diring , Kamel Hadj-Kaddour , Magali Gary-Bobo , et al.
Dalton Transactions, 2021, 50 (13), pp.4583-4592. ⟨10.1039/d0dt03792c⟩
Journal articles hal-03419895v1
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Anti-protozoal and anti-fungal evaluation of 3,5-disubstituted 1,2-dioxolanes

Alexis Pinet , Sandrine Cojean , Linh Thuy Nguyen , Pedro Vásquez-Ocmín , Alexandre Maciuk , et al.
Bioorganic & Medicinal Chemistry Letters, 2021, 47, pp.128196. ⟨10.1016/j.bmcl.2021.128196⟩
Journal articles hal-03320600v1

Structure–Activity Relationships of Human Urotensin II and Related Analogues on Rat Aortic Ring Contraction

Patricia Labarrère , David Chatenet , Jérôme Leprince , Céline Marionneau , Gervaise Loirand , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2003, 18 (2), pp.77-88. ⟨10.1080/1475636031000093507⟩
Journal articles hal-01962785v1

Structure–activity relationships of urotensin II and URP

Jérôme Leprince , David Chatenet , Christophe Dubessy , Alain Fournier , Bruno Pfeiffer , et al.
Peptides, 2008, 29 (5), pp.658-673. ⟨10.1016/j.peptides.2007.08.014⟩
Journal articles istex hal-01972605v1

Design, synthesis, and evaluation of 1-(N-benzylamino)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents

Francis Giraud , Cédric Logé , Fabrice Pagniez , Damien Crepin , Patrice Le Pape , et al.
Bioorganic and Medicinal Chemistry Letters, 2008, 18 (6), pp.1820 - 1824. ⟨10.1016/j.bmcl.2008.02.027⟩
Journal articles istex hal-01689196v1

Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moiety

Nicolas Lebouvier , Fabrice Pagniez , Muriel Duflos , Patrice Le Pape , Young Min Na , et al.
Bioorganic and Medicinal Chemistry Letters, 2007, 17 (13), pp.3686 - 3689. ⟨10.1016/j.bmcl.2007.04.038⟩
Journal articles istex hal-01689197v1

2- and 3-[(Aryl)(azolyl)methyl]indoles as Potential Non-steroidal Aromatase Inhibitors

Marie-Pierre Lézé , Marc Le Borgne , Pascal Marchand , Denis Loquet , Manuela Kogler , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2004, 19 (6), pp.549 - 557. ⟨10.1080/14756360400004631⟩
Journal articles hal-01689238v1

Potential application of plant lipid transfer proteins for drug delivery

Christine Pato , Marc Le Borgne , Guillaume Le Baut , Patrice Le Pape , Didier Marion , et al.
Biochemical Pharmacology, 2001, 62 (5), pp.555 - 560. ⟨10.1016/S0006-2952(01)00708-0⟩
Journal articles istex hal-01689248v1

A 3D-QSAR CoMSIA study on 3-azolylmethylindoles as anti-leishmanial agents

Francis Giraud , Cédric Logé , Marc Le Borgne , Francis Pagniez , Young Min Na , et al.
SAR and QSAR in Environmental Research, 2006, 17 (3), pp.299 - 309. ⟨10.1080/10659360600787494⟩
Journal articles hal-01689291v1

Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1

Espérance Moine , Isabelle Dimier-Poisson , Cécile Enguehard-Gueiffier , Cédric Logé , Mélanie Pénichon , et al.
European Journal of Medicinal Chemistry, 2015, 105, pp.80-105. ⟨10.1016/j.ejmech.2015.10.004⟩
Journal articles hal-02389861v1

Self-assembly of Azacitidine Prodrugs for the Treatment of Myelodysplastic syndromes

Milad Baroud , Olivier Duval , Elise Lepeltier , Yolla El-Makhour , Sylvain Thépot
Association des Enseignants-Chercheurs de Chimie Physique et de Chimie Minérale(AECCPM), Jun 2021, Nantes, France
Conference papers hal-04127323v1
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Heterodimeric Insecticidal Peptide Provides New Insights into the Molecular and Functional Diversity of Ant Venoms

Axel Touchard , Helen Mendel , Isabelle Boulogne , Volker Herzig , Nayara Braga Emidio , et al.
ACS Pharmacology & Translational Science, 2020, 3 (6), pp.1211-1224. ⟨10.1021/acsptsci.0c00119⟩
Journal articles hal-02996356v1
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Two-scale analysis of transient diffusion problems through a homogenized enriched continuum

A. Waseem , T. Heuzé , L. Stainier , M.G.D. G D Geers , V.G. G Kouznetsova
European Journal of Mechanics - A/Solids, 2021, 87, pp.104212. ⟨10.1016/j.euromechsol.2021.104212⟩
Journal articles hal-03164888v1

Synthesis and antileishmanial activity of new imidazolidin-2-one derivatives

Jean-Michel Robert , Caroline Sabourin , Nidia Alvarez , Sylvie Robert-Piessard , Guillaume Le Baut , et al.
European Journal of Medicinal Chemistry, 2003, 38 (7-8), pp.711-718. ⟨10.1016/s0223-5234(03)00119-3⟩
Journal articles istex hal-02389889v1
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Self-assemblies of azacitidine prodrugs: a promising strategy of treatment for myelodysplastic syndromes

Milad Baroud , Elise Lepeltier , Yolla El-Makhour , Sylvain Thépot , Olivier Duval
4th NANOMED EMJMD's workshop (Nanomed 2021), Jul 2021, Angers, France
Conference poster hal-04127352v1

Synthesis and biological evaluation of 3-(azolylmethyl)-1 H -indoles and 3-(α-azolylbenzyl)-1 H -indoles as selective aromatase inhibitors

Marc Le Borgne , Pascal Marchand , Marie-Renée Nourrisson , Denis Loquet , Martina Palzer , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2007, 22 (5), pp.667 - 676. ⟨10.1080/14756360701652658⟩
Journal articles hal-01689199v1
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Phosphonic Acid Fluorescent Organic Nanoparticles for High-Contrast and Selective Staining of Gram-Positive Bacteria

Joanna Boucard , Rym Boudjemaa , Karine K. Steenkeste , Cedric Jacqueline , Nicolas Stephant , et al.
ACS Omega, 2018, 3 (12), pp.17392-17402. ⟨10.1021/acsomega.8b02603⟩
Journal articles hal-02001014v1
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Computational Analysis of Chemical Space of Natural Compounds Interacting with Sulfotransferases

Iglika Lessigiarska , Yunhui Peng , Ivanka Tsakovska , Petko Alov , Nathalie Lagarde , et al.
Molecules, 2021, 26 (21), pp.6360. ⟨10.3390/molecules26216360⟩
Journal articles hal-03448343v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors

Bruno Oyallon , Marie Brachet-Botineau , Cédric Logé , Pascal Bonnet , Mohamed Souab , et al.
European Journal of Medicinal Chemistry, 2018, 154, pp.101-109. ⟨10.1016/j.ejmech.2018.04.056⟩
Journal articles hal-03408667v1
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Study of cytotoxic and photodynamic activities of dyads composed of a zinc phthalocyanine appended to an organotin

Isabelle Toubia , Christophe Nguyen , Stéphane Diring , Marine Pays , Elodie Mattana , et al.
Pharmaceuticals, 2021, 14 (5), ⟨10.3390/ph14050413⟩
Journal articles hal-03419889v1

Thiazolylaminomannosides As Potent Antiadhesives of Type 1 Piliated Escherichia coli Isolated from Crohn’s Disease Patients

Sami Brument , Adeline Sivignon , Tetiana Dumych , Nicolas Moreau , Goedele Roos , et al.
Journal of Medicinal Chemistry, 2013, 56 (13), pp.5395 - 5406. ⟨10.1021/jm400723n⟩
Journal articles hal-01931359v1

Synthetic studies toward the anthrax tetrasaccharide: alternative synthesis of this antigen

Ophélie Milhomme , Sandrine G.Y. Dhénin , Florence Djedaini-Pilard , Vincent Moreau , Cyrille Grandjean
Carbohydrate Research, 2012, 356, pp.115-131. ⟨10.1016/j.carres.2012.01.007⟩
Journal articles istex hal-02196970v1

Synthesis and immunosuppressive activity evaluation of substituted N -imidazolidin-2-ones and N -tetrahydropyrimidin-2(1 H )-ones

Caroline Sabourin , Jean-Michel Robert
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 23 (5), pp.659-667. ⟨10.1080/14756360802205455⟩
Journal articles hal-02389880v1

Straightforward approach to graft bioactive polysaccharides onto polyurethane surfaces using an ionic liquid

Sandra Bigot , Guy Louarn , Nasreddine Kebir , Fabrice Burel
Applied Surface Science, 2014, 314, pp.301-307. ⟨10.1016/j.apsusc.2014.06.114⟩
Journal articles hal-02298991v1

Enhancement of Thermal Conduction of Polyimide/Boron Nitride Nanocomposites

François Saysouk , Sombel Diaham , Marie-Laure Locatelli , B.E. Belkerk , Yves Scudeller , et al.
IEEE Annual Report Conference on Electrical Insulation and Dielectric Phenomena (CEIDP), IEEE, Oct 2013, Shenzhen, China. pp.543-546, ⟨10.1109/CEIDP.2013.6747082⟩
Conference papers hal-02556233v1
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Binding of Gold(III) Porphyrin by the Pro-metastatic Regulatory Protein Human Galectin-3

Vanya Bogoeva , Miroslav Rangelov , Nadezhda Todorova , Annie Lambert , Clarisse Bridot , et al.
Molecules, 2019, 24 (24), pp.4561. ⟨10.3390/molecules24244561⟩
Journal articles hal-02408764v1

Electrochemically promoted tyrosine-click-chemistry for protein labeling

Dimitri Alvarez Dorta , Christine Thobie-Gautier , Mickael Croyal , Mohammed Bouzelha , Mathieu Mevel , et al.
Journal of the American Chemical Society, 2018, ⟨10.1021/jacs.8b09372⟩
Journal articles hal-02621835v1

Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides 2004. Proceedings of the 3rd International and 28th European Symposium, pp 804-805

David Chatenet , Jérôme Leprince , Christophe Dubessy , Ludovic Carlier , Cedric Boularan , et al.
Books hal-01960838v1

The Antiadhesive Strategy in Crohn′s Disease: Orally Active Mannosides to Decolonize Pathogenic Escherichia coli from the Gut

Dimitri Alvarez Dorta , Adeline Sivignon , Thibaut Chalopin , Tetiana Dumych , Goedele Roos , et al.
ChemBioChem, 2016, 17 (10), pp.936-952. ⟨10.1002/cbic.201600018⟩
Journal articles istex hal-02077036v1